2019年度 修了・卒業生
■ 修了生
| Amol D. Sonawane (2017/4-) |
Cascade cyclization and photophysical properties of quinoline/ isoquinoline-based heteroacenes （キノリン/イソキノリン骨格を有するヘテロアセンのカスケード環化と光物理的特性） |
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| Synthesis of thieno[2,3–b]quinoline and selenopheno[2,3–b]quinoline derivatives via iodocyclization reaction and DFT mechanistic study Amol D. Sonawane, Dinesh R. Garud, Taro Udagawa, Mamoru Koketsu Organic & Biomolecular Chemistry, 16(2), 245-255 (2018). |
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| Synthesis of thieno[2,3-c]acridine and furo[2,3-c]acridine derivatives via iodocyclization reaction, fluorescence properties and DFT mechanistic study Amol D. Sonawane, Dinesh R. Garud, Taro Udagawa, Yasuhiro Kubota, Mamoru Koketsu New Journal of Chemistry, 42(18), 15315-15324 (2018). |
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| Synthesis of isoquinoline-fused quinazolinones through Ag(I)-catalyzed cascade annulation of 2-aminobenzamides and 2-alkynylbenzaldehydes Amol D. Sonawane, Yunnus B. Shaikh, Dinesh R. Garud, Mamoru Koketsu Synthesis, 51(2), 500-507 (2019). |
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| Iron-promoted intramolecular cascade cyclization for the synthesis of selenophene-fused, quinoline-based heteroacenes Amol D. Sonawane, Yasuhiro Kubota, Mamoru Koketsu The Journal of Organic Chemistry, 84(13), 8602-8614 (2019). |
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| Iodine mediated in situ generation of R-Se-I: Application towards the construction of pyrano[4,3-b]quinoline heterocycles and fluorescence properties Amol D. Sonawane, Rohini D. Sonawane, Khin Myat Noe Win, Masayuki Ninomiya, Mamoru Koketsu Organic & Biomolecular Chemistry, 17(40), 9039-9049 (2019). |
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| The in-situ air oxidation and photophysical studies of isoquinoline-based N-heteroacenes Khin Myat Noe Win, Amol D. Sonawane, Mamoru Koketsu Organic & Biomolecular Chemistry, 18(11), 2129-2138 (2020). |
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| Synthesis and photophysical properties of selenopheno[2,3-b]quinoxaline and selenopheno[2,3-b]pyrazine heteroacenes Amol D. Sonawane, Atsushi Shimozuma, Taro Udagawa, Masayuki Ninomiya, Mamoru Koketsu Organic & Biomolecular Chemistry, 18, 4063-4070 (2020). |
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| Design and synthesis of quinoxaline-1,3,4-oxadiazole hybrid derivatives as poptent inhibitors of the anti-apoptotic Bcl-2 protein< Yukari Ono, Masayuki Ninomiya, Daiki Kaneko, Amol D. Sonawane, Taro Udagawa, Kaori Tanaka, Atsuyoshi Nishina, Mamoru Koketsu Bioorganic Chemistry, 104, 104245 (2020). |
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| Synthesis of [1,2,4]triazolo[4,3-a]quinoxaline-1,3,4-oxadiazole derivatives as potent antiproliferative agents via a hybrid pharmacophore approach Daiki Kaneko, Masayuki Ninomiya, Rina Yoshikawa, Yukari Ono, Amol D. Sonawane, Kaori Tanaka, Atsuyoshi Nishina, Mamoru Koketsu Bioorganic Chemistry, 104, 104293 (2020). |
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| Synthesis of selenated tetracyclic indoloazulenes via iodine and diorganyl diselenides Khin Myat Noe Win, Amol D. Sonawane, Mamoru Koketsu Organic & Biomolecular Chemistry, in press | |
| Synthesis of organoselenium scaffolds through selenium radical formation Amol D. Sonawane, Mamoru Koketsu in Organoselenium Chemistry, Brindaban C. Ranu, Bubun Banerjee Eds., Walter de Gruyter GmbH, Berlin, Germany, 2020 Chapter 2, pp. 29-53. |
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| Role of isoselenocyanates for the synthesis of selenium-containing heterocycles Amol D. Sonawane, Mamoru Koketsu in Organoselenium Chemistry, Brindaban C. Ranu, Bubun Banerjee Eds., Walter de Gruyter GmbH, Berlin, Germany, 2020 Chapter 3, pp. 55-83. |
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| Recent advances on C-Se Bond-forming reactions at low and room temperature Amol D. Sonawane, Mamoru Koketsu Current Organic Chemistry, 23(2), 3206-3225 (2019). |
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| Synthesis of Se-heterocycles by cascade cyclization of heteroatom containing alkynes Amol D. Sonawane, Rohini A. Sonawane, Masayuki Ninomiya, Mamoru Koketsu Advances Synthesis & Catalysis, 362, 3485-3515 (2020). |
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| Organocatalysed synthesis of selenium containing scaffolds Amol D. Sonawane,Mamoru Koketsu Current Organocatalysis, 8(1), 5-26 (2021). |
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| 大野 友花里 (2017/4-) |
抗アポトーシス性タンパク質Bcl-2を標的としたキノキサリン誘導体の合成 |
| Design and synthesis of quinoxaline-1,3,4-oxadiazole hybrid derivatives as poptent inhibitors of the anti-apoptotic Bcl-2 protein< Yukari Ono, Masayuki Ninomiya, Daiki Kaneko, Amol D. Sonawane, Taro Udagawa, Kaori Tanaka, Atsuyoshi Nishina, Mamoru Koketsu Bioorganic Chemistry, 104, 104245 (2020). |
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| Synthesis of [1,2,4]triazolo[4,3-a]quinoxaline-1,3,4-oxadiazole derivatives as potent antiproliferative agents via a hybrid pharmacophore approach Daiki Kaneko, Masayuki Ninomiya, Rina Yoshikawa, Yukari Ono, Amol D. Sonawane, Kaori Tanaka, Atsuyoshi Nishina, Mamoru Koketsu Bioorganic Chemistry, 104, 104293 (2020). |
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| 兼子 大輝 (2017/4-) |
イミカリン誘導体の合成とそれらのヒトガン細胞に対する細胞毒性の検討 |
| Design and synthesis of quinoxaline-1,3,4-oxadiazole hybrid derivatives as poptent inhibitors of the anti-apoptotic Bcl-2 protein< Yukari Ono, Masayuki Ninomiya, Daiki Kaneko, Amol D. Sonawane, Taro Udagawa, Kaori Tanaka, Atsuyoshi Nishina, Mamoru Koketsu Bioorganic Chemistry, 104, 104245 (2020). |
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| Synthesis of [1,2,4]triazolo[4,3-a]quinoxaline-1,3,4-oxadiazole derivatives as potent antiproliferative agents via a hybrid pharmacophore approach Daiki Kaneko, Masayuki Ninomiya, Rina Yoshikawa, Yukari Ono, Amol D. Sonawane, Kaori Tanaka, Atsuyoshi Nishina, Mamoru Koketsu Bioorganic Chemistry, 104, 104293 (2020). |
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| 下妻 篤史 (2017/4-) |
セレノフェノキノキサリン誘導体の合成とAChE阻害能の検討 |
| Synthesis and photophysical properties of selenopheno[2,3-b]quinoxaline and selenopheno[2,3-b]pyrazine heteroacenes Amol D. Sonawane, Atsushi Shimozuma, Taro Udagawa, Masayuki Ninomiya, Mamoru Koketsu Organic & Biomolecular Chemistry, 18, 4063-4070 (2020). |
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| 杉山 穂高 (2017/4-) |
テルフェニルキノン誘導体の合成とヒト白血病細胞に対する細胞毒性の評価 |
■ 卒業生
| 岡部 紗世 (2019/4-) |
フラボノイド類縁体の合成とそれらのアセチルコリンエステラーゼ阻害能に関する比較研究 |
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| 吉川 利奈 (2019/4-) |
イミキモド誘導体の化学修飾とガン細胞に対する細胞毒性評価 |