2001年度 修了・卒業生 (石原研)
■ 修了生
| 加納 征典 (1999/4-) | アルキンセレノラートとジフェニルケテンの反応による[2+2]環化付加を介した3-アルキルセレノ-2-シクロブテノンの簡便な合成法 |
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| Synthesis of 1-alkylselenocyclobutene via intermediate allenyl selenoketene M. Koketsu, M. Kanoh, Y. Yamamura, H. Ishihara Tetrahedron Lett., 46, 1479-1481 (2005). |
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| Reactions of 2-pentynyl trimethylsilylethynyl selenides with primary amines via allenyl selenoketene M. Koketsu, M. Kanoh, H. Ishihara J. Heterocycl. Chem., 42, 293-296 (2005). |
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| Synthesis of 3-alkylseleno-2-cylcobutenone via [2+2]cycloaddition reaction of alkyneselenolate with diphenylketene M. Koketsu, M. Kanoh, H. Ishihara Synlett, 805-807 (2002). |
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| Reaction of allenyl selenoketene, generated by [3,3] sigmatropic rearrangement, with amines M. Koketsu, M. Kanoh, E. Itoh, H. Ishihara J. Org. Chem., 66, 4099-4101 (2001). |
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| 竹中 雄一 (1999/4-) | 第一セレノアミドを用いた含セレン環状化合物の合成 |
| Syntheses of cyanoselenoamides and diselenoamides. Their conversion into selenazole and selenazine M. Koketsu, Y. Takenaka, H. Ishihara Heteroatom Chem., 14, 106-110 (2003). |
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| Synthesis of 1,3-thiazine derivatives as potential antimycobacterial agents M. Koketsu, K. Tanaka, Y. Takenaka, C. D. Kwong, H. Ishihara Eur. J. Pharm. Sci., 15, 307-310 (2002). |
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| Facile preparation of 1,3-selenazine derivatives by reaction of primary selenoamides with α,β-unsaturated aldehydes of in the presence of BF3 ･Et2O M. Koketsu, Y. Takenaka, S. Hiramatsu, H. Ishihara Heterocycles, 55, 1181-1188 (2001). |
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| Preparation of 1,3-selenazol-4-one derivatives from primary selenoamides and haloacyl halides M. Koketsu, Y. Takenaka, H. Ishihara Synthesis, 731-734 (2001). |
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| 名田 大志 (1999/4-) | LiAlHSeHを用いたセレン化合物の合成および含セレン環状化合物合成反応の開発 |
| Synthesis of 4-selenazolones. Hetero Diels-Alder reaction of selenazadienes with DMAD M. Koketsu, F. Nada, T. Mio, H. Ishihara Heterocycles, 60, 1211-1218 (2003). |
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| Facile preparation of 2-imino-1,3-selenazolidin-4-one derivatives by reaction of selenoureas with a -haloacyl halides M. Koketsu, F. Nada, H. Ishihara Synthesis, 195-198 (2002). |
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| Reactions of acyl chlorides with LiAlHSeH. Preparation of diacyl selenides, diacyl diselenides, selenocarboxylates and cyclic selenoanhydrides M. Koketsu, F. Nada, S. Hiramatsu, H. Ishihara J. Chem. Soc. Perkin Trans., 1, 737-740 (2002). |
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| Reaction of lithium aluminium hydride with elemental selenium. Its application as a selenating reagent into organic molecules H. Ishihara, M. Koketsu, Y. Fukuta, F. Nada J. Am. Chem. Soc., 123, 8408-8409 (2001). |
■ 卒業生
| 小林 親司 (2001/4-) | LiAlHSHを用いたチオカルバミン酸エステルの合成 |
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| Synthesis of N-aryl S-alkylthiocarbamates M. Koketsu, C. Kobayashi, H. Ishihara Heteroatom Chem., 14, 374-378 (2003). |
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| 桜井 久子 (2001/4-) | 抗カビ作用を有するフラボノイド3糖の合成を目指した研究 |
| First synthesis of a trisaccharide of glycosylkaemferide: A resistance factor in carnationss M. Koketsu, M. Kuwahara, H. Sakurai, H. Ishihara Synthetic Commun., 34, 239-245 (2004). |
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| 中島 世津子 (2001/4-) | セレノ尿素を用いたベンゾセレナゾールの合成 |